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Microsatellite instable cancer cells acquire on-target resistance mutations to WRN helicase inhibitors

Faith Fowler, Jessica Gajda, Amirhossein Mafi, Aileen Kelly, Cynthia L Jeffries, Phuong Le, Lei Shi, Mariam George, Nathaniel Elsen, Alla V Korepanova, Sarah M Zerbs, Orville A Pemberton, Xiangdong Xu, Nathan Gesmundo, Wei Qiu, Fei Han, Henry Tang, Sanjay C Panchal, Michael Dart, Jonathan Hickson, Chaohong Sun, Yunsong Tong, Ari J Firestone
Molecular Cancer Therapeutics February 9, 2026