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Discovery of Fosigotifator, a Potent eIF2B Activator with Desired Properties for Human Studies

Jennifer M Frost, Yunsong Tong, Xiangdong Xu, Lei Shi, Marina Pliushchev, Kathleen J Murauski, Kathy Kohlhaas, Diana L Donnelly-Roberts, Michael M Sheehan, Stephan Riedmaier, Hardeep S Oberoi, Jun Chen, Janani Prakash, Charles W Hutchins, Clarissa G Jakob, Rinku Jain, Wei Qiu, Rodger F Henry, Rohinton Edalji, Chaohong Sun, Tracy Carr, Ana M Basso, Brian S Brown, Eric A Voight, Carmela Sidrauski, Michael J Dart
Journal of Medicinal Chemistry May 19, 2026